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Submit ReviewElinogrel
Description: P2Y12 antagonist
Chemical Name: 5-Chloro-N-[[[4-[6-Fluoro-1,4-dihydro-7-(methylamino)-2,4-dioxo-3(2H)-quinazolinyl]phenyl]amino]carbonyl]-2-thiophenesulfonamide
Purity: ≥97% (HPLC)
Biological Activity for Elinogrel
Elinogrel is a P2Y12 antagonist; exhibits antiplatelet activity.
Compound Libraries for Elinogrel
Elinogrel is also offered as part of the Tocriscreen 2.0 Max. Find out more about compound libraries available from Tocris.
Technical Data for Elinogrel
| M. Wt | 523.95 |
| Formula | C20H15ClFN5O5S2 |
| Storage | Store at -20°C |
| Purity | ≥97% (HPLC) |
| CAS Number | 936500-94-6 |
| PubChem ID | 16066663 |
| InChI Key | LGSDFTPAICUONK-UHFFFAOYSA-N |
| Smiles | O=C(NS(C4=CC=C(Cl)S4)(=O)=O)NC(C=C3)=CC=C3N2C(C1=CC(F)=C(NC)C=C1NC2=O)=O |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Solubility Data for Elinogrel
| Solvent | Max Conc. mg/mL | Max Conc. mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 52.4 | 100 |
Preparing Stock Solutions for Elinogrel
The following data is based on the product molecular weight 523.95. Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.91 mL | 9.54 mL | 19.09 mL |
| 5 mM | 0.38 mL | 1.91 mL | 3.82 mL |
| 10 mM | 0.19 mL | 0.95 mL | 1.91 mL |
| 50 mM | 0.04 mL | 0.19 mL | 0.38 mL |
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Product Datasheets for Elinogrel
References for Elinogrel
References are publications that support the biological activity of the product.
Cattaneo et al (2010) State of the art of new P2Y12 antagonists. Intern.Emerg.Med. 5 385 PMID: 20177818
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Keywords: Elinogrel, Elinogrel supplier, P2Y12, receptor, antagonists, antiplatelet, antagonises, inhibitors, inhibits, Purinergic, P2Y, Receptors, 5316, Tocris Bioscience
1 Citation for Elinogrel
Citations are publications that use Tocris products. Selected citations for Elinogrel include:
Tuan et al (2021) A small molecule UPR modulator for diabetes identified by high throughput screening. Acta Pharm Sin B 11 3983-3993 PMID: 35024320
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Literature in this Area
Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* your copy today!
*Please note that Tocris will only send literature to established scientific business / institute addresses.
P2X and P2Y Receptors Scientific Review
Written by Kenneth Jacobson, this review provides an overview of the different subtypes and structures of the P2 receptor families, as well as the pharmacological probes used to study them; compounds available from Tocris are listed.